Orexin Circuit & Dual Receptor Dynamics

Hypothalamic OX1R/OX2R Flip-Flop Neuromorphic Simulator

OX2R Agonist Mode
Lateral Hypothalamus → Brainstem Circuit Wake Firing: 18.6 Hz
Flip-Flop State Trajectory & Membrane Excitability Bistable Attractor
Receptor Occupancy & Flip-Flop Balance Danavorexton / TAK-861 Class
FLIP-FLOP STATE: STABLE ACTIVE WAKE
OX2R Occupancy
91.4%
OX1R Occupancy
4.2%
Wake Firing Rate
18.6 Hz
Cataplexy Vulnerability
0.12
NREM Latency
420 min
VLPO GABA Drive
0.65
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